商品名(trade name) | |
藥理作用(Pharmacological Effects) | [hyperpolarization: increase ATP-sensitive K+ channels-->K+ exflux [causes local relaxation in smooth muscle by increasing membrane permeability to potassium ions-->smooth muscle hard to reach threshold-->vasodialation [Ca2+ influx decrease-->contraction of smooth muscle decrease [no diuretic effect |
用量與用法(Dosage and Usage) | usage ]IV ]unchanged form urine excretion |
適應症(Indications) | {acute hypertension: vasodilator {malignant hypertension: vasodilator {Insulinoma(胰島細胞瘤): could reduce insulin secretion {ongenital hyperinsulinism: could reduce insulin secretion |
副作用(Side effect) | }Coronary and cerebral vascular insufficiency }diabetes mellitus(糖尿病): ATP-sensitive K+ channels, and beta cell at pancreas will hyperpolarization }Compensatory edema: due to vasodilation |
禁忌/交互作用(Contraindications / interaction) |
Monday, October 21, 2013
diazoxide
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