Monday, November 11, 2013

procainamide

商品名(trade name)

藥理作用(Pharmacological Effects)
[more stable and less central action than quinidine
[heart: like quinidine
[ANS: M receptor block is weak and no alpha receptor inhibition
用量與用法(Dosage and Usage)
usage
]per os, IM, IV (prn)
Pharmacokinetics
]Well absorbed
]20 % plasma protein binding,
]t1/2=5~8 hours
適應症(Indications)
{like quinidine
副作用(Side effect)
}predominant lupus like syndrome: slow acetylator, accumulate too much drug in body and cannot be metabolic by liver
}G-I disturbance: less common than quinidine
}Cardiotoxicity: can produce paradoxical ventricular tachycardia (Torsade de pointes)
}lupus like syndrome
禁忌/交互作用(Contraindications / interaction)

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